SCHEMBL5260346

SCHEMBL5260346

CC(c1ccc(Cl)cc1)C(CNC(=O)c1cccc(N2CCNC2=O)c1)c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.46
NPC1 O15118 2/20 0.46
ITGB3 P05106 1/20 0.40
ITGB1 P05556 1/20 0.40
ITGAV P06756 1/20 0.40
ITGA5 P08648 1/20 0.40
ITGA4 P13612 1/20 0.40
ITGB5 P18084 1/20 0.40
ITGB8 P26012 1/20 0.40
KMT2A Q03164 5/20 0.39
GAA P10253 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TP53 P04637 2/20 0.38
MEN1 O00255 2/20 0.38
LMNA P02545 1/20 0.38
CYP24A1 Q07973 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HCRTR1 O43613 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5263063 0.85 RAB9A (0.65) RAB9ANPC1KMT2AGAAMEN1
SCHEMBL5260117 0.81 CNR1 (0.54) RAB9ANPC1CNR1CNR2
SCHEMBL3237117 0.81 NPC1 (0.56) RAB9ANPC1KMT2AMEN1LMNA
SCHEMBL4688879 0.80 MAPT (0.43) RAB9ANPC1ITGB3ITGB1ITGAV
SCHEMBL5264039 0.79 KMT2A (0.53) RAB9ANPC1KMT2AGAAHSD17B10
SCHEMBL5259145 0.76 ALDH1A1 (0.46) RAB9ANPC1KMT2AGAAHSD17B10
SCHEMBL5262774 0.75 SLC6A9 (0.54) RAB9ANPC1KMT2AGAAHSD17B10
SCHEMBL5266049 0.73 RAB9A (0.60) RAB9ANPC1KMT2ATP53MEN1
SCHEMBL5263349 0.72 MAPT (0.65) RAB9ANPC1KMT2AHSD17B10MEN1
SCHEMBL5262488 0.71 SLC6A9 (0.55) RAB9ANPC1KMT2AMEN1CYP24A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP disclosed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP disclosed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO disclosed