SCHEMBL5259209

SCHEMBL5259209

CCC#Cc1cccc(CF)n1

nearest known ligand 0.42

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 14/20 0.41
TRPV3 Q8NET8 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347186 0.82 GRM5 (0.37) GRM5TRPV3
SCHEMBL103337 0.79 GRM5 (0.42) GRM5TRPV3
SCHEMBL103656 0.79 GRM5 (0.42) GRM5TRPV3
SCHEMBL103768 0.79 CHRNB2 (0.43) GRM5TRPV3
SCHEMBL5258543 0.77 GRM5 (0.66) GRM5
SCHEMBL14207818 0.74 GRM5 (0.42) GRM5
SCHEMBL101806 0.74 GRM5 (0.38) GRM5
SCHEMBL28020770 0.73 CTSS (0.40)
SCHEMBL3354041 0.73 KCNH2 (0.33)
SCHEMBL102431 0.72 GRM5 (0.48) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765795-A2 ALKYNYL DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS Addex Pharmaceuticals SA (CH) 2007-03-28 EP disclosed
WO-2005123703-A2 ALKYNYL DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX PHARMACEUTICALS SA (CH) 2005-12-29 WO disclosed