SCHEMBL525922

SCHEMBL525922

C=CCc1ccc(O)c(-c2cc(CC=C)ccc2OC(=O)C(CCC)CCC)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 9/20 0.60
GABRB2 P47870 9/20 0.60
CNR2 P34972 4/20 0.54
CNR1 P21554 3/20 0.54
ALDH1A1 P00352 2/20 0.54
MEN1 O00255 2/20 0.54
GAA P10253 2/20 0.54
MAPT P10636 2/20 0.54
KMT2A Q03164 2/20 0.54
KDM4E B2RXH2 1/20 0.54
ALDH2 P05091 1/20 0.54
AKR1B1 P15121 1/20 0.54
HPGD P15428 1/20 0.54
PPARG P37231 1/20 0.54
PPARD Q03181 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
TNKS O95271 1/20 0.50
PARP1 P09874 1/20 0.50
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4744358 0.79 GABRA1 (0.63) GABRA1GABRB2CNR2CNR1ALDH1A1
Hydrochloric Acid SCHEMBL4742209 0.78 GABRA1 (0.61) GABRA1GABRB2CNR2CNR1ALDH1A1
SCHEMBL724850 0.77 NOS2 (0.44) MEN1KMT2ACYP3A4
Hydrochloric Acid SCHEMBL530776 0.77 NOS2 (0.44) MEN1KMT2ACYP3A4
SCHEMBL525807 0.76 GABRA1 (0.74) GABRA1GABRB2CNR2CNR1ALDH1A1
SCHEMBL525761 0.76 GABRA1 (1.00) GABRA1GABRB2CNR2CNR1ALDH1A1
SCHEMBL31051046 0.75 GABRA1 (0.60) GABRA1GABRB2CNR2CNR1ALDH1A1
SCHEMBL18313945 0.74 ALOX5 (0.75) GABRA1GABRB2CNR2CNR1ALDH1A1
SCHEMBL22215973 0.74 GABRA1 (0.89) GABRA1GABRB2CNR2CNR1ALDH1A1
Magnolol SCHEMBL23119980 0.73 GABRA1 (0.85) GABRA1GABRB2CNR2CNR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP disclosed
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP disclosed
WO-2012013691-A1 MULTITARGET SUBSTITUTED BIPHENYL DIOL DERIVATIVES PROUS INSTITUTE FOR BIOMEDICAL RESEARCH, S.A. (ES) 2012-02-02 WO disclosed
WO-2012013691-A1 MULTITARGET SUBSTITUTED BIPHENYL DIOL DERIVATIVES PROUS INSTITUTE FOR BIOMEDICAL RESEARCH, S.A. (ES) 2012-02-02 WO disclosed