SCHEMBL5264063

SCHEMBL5264063

CC(c1ccc(Cl)cc1)C(CNC(=O)c1cccc2ccncc12)c1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.44
BAD Q92934 2/20 0.44
PIM2 Q9P1W9 2/20 0.44
P2RX7 Q99572 10/20 0.42
PREP P48147 1/20 0.41
HDAC2 Q92769 1/20 0.39
TRPV1 Q8NER1 2/20 0.39
DGAT2 Q96PD7 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5262202 0.92 TRPV1 (0.45) PIM1BADPIM2P2RX7PREP
SCHEMBL5367653 0.87 P2RX7 (0.49) P2RX7HDAC2NPC1RAB9A
SCHEMBL5261775 0.80 NSD2 (0.52) P2RX7
SCHEMBL5264060 0.80 CNR1 (0.49)
SCHEMBL5262392 0.78 SLC6A9 (0.53) RAB9A
SCHEMBL5261739 0.77 NPC1 (0.61) P2RX7NPC1RAB9A
SCHEMBL5262488 0.77 SLC6A9 (0.55) P2RX7NPC1RAB9A
SCHEMBL5262900 0.77 NSD2 (0.45) P2RX7PREP
SCHEMBL5261415 0.76 P2RX7 (0.46) P2RX7NPC1RAB9A
SCHEMBL5264103 0.76 CYP1A2 (0.58) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP disclosed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP disclosed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO disclosed