SCHEMBL5266002

SCHEMBL5266002

CC(=O)Nc1c[nH]nc1C(=O)NC(C)C

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.42
CYP1A2 P05177 1/20 0.42
KDM4E B2RXH2 2/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
DYRK1A Q13627 4/20 0.36
MLYCD O95822 1/20 0.35
ALDH1A1 P00352 3/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 2/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13816853 0.83 SMN1; SMN2 (0.44) SMN1; SMN2CYP1A2KDM4EADORA3ADORA2A
SCHEMBL2801403 0.83 HSD17B10 (0.38) KDM4EADORA3ALDH1A1RAB9ALMNA
SCHEMBL5269232 0.81 CLK1 (0.49) PKMTSHR
SCHEMBL5267481 0.81 MDM4 (0.49) SMN1; SMN2CYP1A2ADORA3ADORA2AADORA2B
SCHEMBL5270659 0.80 KDM4E (0.44) SMN1; SMN2CYP1A2KDM4EALDH1A1RAB9A
SCHEMBL23844229 0.79 SMN1; SMN2 (0.43) SMN1; SMN2CYP1A2KDM4EADORA3ADORA2A
SCHEMBL5268520 0.79 ALDH1A1 (0.47) SMN1; SMN2KDM4EALDH1A1RAB9ALMNA
SCHEMBL5269964 0.79 HTT (0.50) SMN1; SMN2KDM4EALDH1A1RAB9ALMNA
SCHEMBL5269326 0.78 KDM4E (0.42) SMN1; SMN2CYP1A2KDM4EADORA3ADORA2A
SCHEMBL5268963 0.78 LMNA (0.46) SMN1; SMN2CYP1A2ALDH1A1PKMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed