SCHEMBL5266987

SCHEMBL5266987

CC1(C)C=C(C#N)c2cc(F)c(Cl)cc2OC1

nearest known ligand 0.36

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.36
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5271209 0.89
SCHEMBL5273430 0.78 PGR (0.37) NOTUM
SCHEMBL5271201 0.78 PGR (0.37) NOTUMAKR1B1
SCHEMBL1400074 0.76 NOTUM (0.36) NOTUMAKR1B1
SCHEMBL5269873 0.75 ALDH1A1 (0.37)
SCHEMBL5269692 0.72 NR3C1 (0.37)
SCHEMBL5559796 0.72 NOTUM (0.31) NOTUMAKR1B1
SCHEMBL5270297 0.71 OPRD1 (0.35)
SCHEMBL2317446 0.70 NOTUM (0.37) NOTUMAKR1B1
SCHEMBL2317447 0.70 NOTUM (0.37) NOTUMAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1600446-B1 New 3,3-dimethyl-5-cyano-benzoxepine derivatives useful for the preparation of 5-formyl-benzoxepine derivatives MERCK SANTE SAS (FR) 2007-10-17 EP claimed
EP-1600446-A1 New 3,3-dimethyl-5-cyano-benzoxepine derivatives useful for the preparation of 5-formyl-benzoxepine derivatives Merck Sante (FR) 2005-11-30 EP claimed
WO-2005111012-A1 NEW 3,3-DIMETHYL-5-CYANO-BENZOXEPINES DERIVATIVES USEFUL FOR THE PREPARATION OF 5-FORMYL-BENZOXEPINE DERIVATIVES MERCK PATENT GMBH (DE) 2005-11-24 WO claimed
EP-1600446-B1 New 3,3-dimethyl-5-cyano-benzoxepine derivatives useful for the preparation of 5-formyl-benzoxepine derivatives MERCK SANTE SAS (FR) 2007-10-17 EP disclosed
EP-1600446-A1 New 3,3-dimethyl-5-cyano-benzoxepine derivatives useful for the preparation of 5-formyl-benzoxepine derivatives Merck Sante (FR) 2005-11-30 EP disclosed
WO-2005111012-A1 NEW 3,3-DIMETHYL-5-CYANO-BENZOXEPINES DERIVATIVES USEFUL FOR THE PREPARATION OF 5-FORMYL-BENZOXEPINE DERIVATIVES MERCK PATENT GMBH (DE) 2005-11-24 WO disclosed