SCHEMBL5276396

SCHEMBL5276396

COc1cc2c(cc1OC)CN(CCC(=O)NCCC(c1ccccc1)c1ccccc1)C(C)C2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.52
ADRA2B P18089 1/20 0.52
ADRA2C P18825 1/20 0.52
ADRA1D P25100 1/20 0.52
ADRA1A P35348 1/20 0.52
ADRA1B P35368 1/20 0.52
MTNR1A P48039 5/20 0.48
MTNR1B P49286 5/20 0.48
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
AGTR2 P50052 1/20 0.41
ALOX12 P18054 3/20 0.40
ALDH1A1 P00352 2/20 0.40
HTT P42858 2/20 0.40
KDM4E B2RXH2 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPT P10636 1/20 0.40
RECQL P46063 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5242061 0.81 KMT2A (0.53) MTNR1AMTNR1BKMT2AHCRTR2
SCHEMBL5454057 0.80 ABCB1 (0.54) MEN1KMT2AALDH1A1HTTKDM4E
SCHEMBL5241961 0.80 ADRA2A (0.45) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL5786435 0.72 GPR183 (0.51) KMT2AAGTR2ACE
SCHEMBL5789193 0.71 CA2 (0.41) ADRA1DADRA1BALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL7854656 0.71 DRD2 (0.42) MEN1KMT2AALDH1A1KDM4ELMNA
SCHEMBL5466197 0.71 MTNR1A (0.50) MTNR1AMTNR1BKDM4ECASR
SCHEMBL5786442 0.71 HDAC6 (0.46)
SCHEMBL5276997 0.70 CA2 (0.45) KMT2AAGTR2ALDH1A1KDM4E
SCHEMBL10974666 0.69 ADRA2A (0.98) ADRA2AADRA2BADRA2CADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833797-A1 AZACYCLIC COMPOUNDS AS INHBITORS OF SENSORY NEURONE SPECIFIC CHANNELS (SNS) VERNALIS (R&D) LTD (GB) 2007-09-19 EP disclosed
WO-2006082354-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC CHANNELS ( SNS ) VERNALIS (R & D) LIMITED (GB) 2006-08-10 WO disclosed