SCHEMBL5280054

SCHEMBL5280054

CCOC(=O)Oc1cnc(-c2ccc(C)c(F)c2)nc1Oc1cc(Cl)ccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
GAA P10253 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
CYP1A2 P05177 4/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
POLB P06746 2/20 0.39
GPBAR1 Q8TDU6 2/20 0.38
GABRA2 P47869 2/20 0.36
GABRB2 P47870 2/20 0.36
SCN9A Q15858 5/20 0.36
HTT P42858 1/20 0.36
TSPO P30536 1/20 0.35
ALDH1A1 P00352 1/20 0.35
FOS P01100 1/20 0.34
JUN P05412 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5281504 0.90 MAPT (0.46) MAPTNPSR1GAAGPR55L3MBTL1
SCHEMBL5289303 0.89 L3MBTL1 (0.45) GAAL3MBTL1CYP1A2CYP2C9CYP2C19
SCHEMBL5126518 0.86 CYP1A2 (0.56) MAPTNPSR1GAAGPR55L3MBTL1
SCHEMBL5278083 0.83 ALDH1A1 (0.39) MAPTCYP1A2CYP2C9CYP2C19POLB
SCHEMBL5114037 0.82 TDP1 (0.50) L3MBTL1CYP1A2CYP2C9CYP2C19POLB
SCHEMBL5282772 0.82 L3MBTL1 (0.56) MAPTNPSR1GAAGPR55L3MBTL1
SCHEMBL5289551 0.81 MAPT (0.48) MAPTNPSR1GAAGPR55L3MBTL1
SCHEMBL5296815 0.81 MAPT (0.48) MAPTNPSR1GAAGPR55L3MBTL1
SCHEMBL5287033 0.81 LMNA (0.45) MAPTNPSR1GAAGPR55L3MBTL1
SCHEMBL5283873 0.80 MAPT (0.47) MAPTNPSR1GAAGPR55L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1866289-A1 PYRIMIDINE CARBOXYLIC ACID DERIVATIVES AND USE THEREOF Bayer HealthCare AG (DE) 2007-12-19 EP disclosed
WO-2006097220-A1 PYRIMIDINE CARBOXYLIC ACID DERIVATIVES AND USE THEREOF BAYER HEALTHCARE AG (DE) 2006-09-21 WO disclosed