SCHEMBL5280628

SCHEMBL5280628

O=C(c1ccc(F)cc1NCCc1cc(Cl)cc(Cl)c1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.39
ACLY P53396 4/20 0.38
MDM2 Q00987 1/20 0.36
RPS6KB1 P23443 3/20 0.35
AKT1 P31749 3/20 0.35
MARS1 P56192 1/20 0.34
IDO1 P14902 1/20 0.34
HPGD P15428 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1748251 0.87 ACLY (0.50) ACLYMDM2RPS6KB1MARS1IDO1
SCHEMBL5275083 0.85 HDAC3 (0.48) ALDH1A1MEN1LMNAHTTKMT2A
SCHEMBL5274599 0.82 CNR1 (0.40) CNR1MEN1HTTKMT2ASMN1; SMN2
SCHEMBL5272631 0.78 HTR6 (0.46) ALDH1A1HTT
SCHEMBL5280864 0.73 SMN1; SMN2 (0.47) ALDH1A1MEN1LMNAHTTKMT2A
SCHEMBL1748139 0.72 GRN (0.36) ACLYMDM2ALDH1A1MEN1KMT2A
SCHEMBL5273090 0.72 CCR2 (0.48) ACLY
SCHEMBL5276755 0.72 CDC7 (0.45) RPS6KB1IDO1HTTHDAC4
SCHEMBL1748141 0.69 AURKA (0.44) RPS6KB1ALDH1A1MEN1HTTKMT2A
SCHEMBL21722883 0.68 HPGD (0.50) HPGDALDH1A1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856075-A1 SUBSTITUTED ARYLAMINE COMPOUNDS AND THEIR USE AS 5-HT6 MODULATORS Epix Delaware, Inc. (US) 2007-11-21 EP disclosed
WO-2006081332-A1 SUBSTITUTED ARYLAMINE COMPOUNDS AND THEIR USE AS 5-HT6 MODULATORS EPIX DELAWARE, INC. (US) 2006-08-03 WO disclosed