SCHEMBL5275083

SCHEMBL5275083

O=C(c1ccc(F)cc1NCCc1ccccc1)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
MLYCD O95822 3/20 0.48
RXFP1 Q9HBX9 1/20 0.46
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 4/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ASPH Q12797 1/20 0.45
RIOX2 Q8IUF8 1/20 0.45
KDM8 Q8N371 1/20 0.45
RAB9A P51151 3/20 0.45
NPC1 O15118 1/20 0.45
KDM6B O15054 1/20 0.44
KDM4C Q9H3R0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5280628 0.85 CNR1 (0.39) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL6719405 0.82 RAB9A (0.64) HDAC3HDAC1MLYCDALDH1A1KDM4E
SCHEMBL5274599 0.82 CNR1 (0.40) HDAC3HDAC4HDAC1HDAC6KDM4E
SCHEMBL4137576 0.77 HTR6 (0.60) RXFP1ALDH1A1POLBMAPTHTR6
SCHEMBL5276755 0.76 CDC7 (0.45) HDAC4RXFP1HTTNPC1MAPT
SCHEMBL7006284 0.74 GRIK1 (0.44) HDAC1ALDH1A1HTTSMN1; SMN2RAB9A
SCHEMBL1748251 0.74 ACLY (0.50) MAPT
SCHEMBL8368711 0.73 RAB9A (0.52) HDAC3HDAC1ALDH1A1KDM4EMEN1
SCHEMBL7835892 0.72 RAB9A (0.57) ALDH1A1KDM4EMEN1KMT2ALMNA
SCHEMBL4217232 0.72 KDM6B (0.61) HDAC6ALDH1A1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856075-A1 SUBSTITUTED ARYLAMINE COMPOUNDS AND THEIR USE AS 5-HT6 MODULATORS Epix Delaware, Inc. (US) 2007-11-21 EP disclosed
WO-2006081332-A1 SUBSTITUTED ARYLAMINE COMPOUNDS AND THEIR USE AS 5-HT6 MODULATORS EPIX DELAWARE, INC. (US) 2006-08-03 WO disclosed