SCHEMBL5281219

SCHEMBL5281219

CC(NC(=O)C1CN(C(=O)c2cccnc2)CCN1)c1cccs1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
MAPK1 P28482 3/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 2/20 0.43
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CASP3 P42574 1/20 0.41
CTSK P43235 1/20 0.41
CTSF Q9UBX1 1/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA7 P36544 1/20 0.41
CHRNA4 P43681 1/20 0.41
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5281221 0.78 CTSL (0.51) ALDH1A1KMT2ACTSLCTSBCASP3
SCHEMBL5191441 0.73 CTSL (0.44) ALDH1A1MAPK1CYP2C19KMT2ALMNA
SCHEMBL5192047 0.69 KMT2A (0.45) ALDH1A1MAPK1CYP2C19KMT2ACTSL
SCHEMBL5192050 0.68 CTSL (0.47) ALDH1A1KMT2ACTSLCTSBCASP3
SCHEMBL5190965 0.66 CHRNB2 (0.51) ALDH1A1MAPK1KMT2ACHRNB2CHRNB4
SCHEMBL29831536 0.65 MKNK1 (0.72) ALDH1A1MAPK1KMT2ACHRNB2CHRNB4
SCHEMBL1088707 0.65 MKNK1 (0.72) ALDH1A1MAPK1KMT2ACHRNB2CHRNB4
SCHEMBL18705009 0.65 MAPK1 (0.64) ALDH1A1MAPK1KMT2AMEN1POLB
SCHEMBL3933150 0.65 GRIN2B (0.46) ALDH1A1CYP2C19KMT2ALMNAITGB3
Hydrochloric Acid SCHEMBL9785721 0.64 MKNK1 (0.70) ALDH1A1MAPK1KMT2ACHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed