SCHEMBL5282643

SCHEMBL5282643

NC(=O)Cc1cccc(Oc2ccncc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.48
FFAR1 O14842 2/20 0.45
CCR8 P51685 1/20 0.45
KCNH2 Q12809 1/20 0.45
BRS3 P32247 1/20 0.44
FAAH O00519 2/20 0.43
TNKS O95271 1/20 0.43
PARP15 Q460N3 1/20 0.43
PARP14 Q460N5 1/20 0.43
PARP10 Q53GL7 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
RAF1 P04049 1/20 0.42
PTGES O14684 1/20 0.42
CYP19A1 P11511 1/20 0.42
ROCK1 Q13464 5/20 0.42
PRKACA P17612 4/20 0.42
CYP3A4 P08684 2/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1395777 0.87 FFAR1 (0.56) F10FFAR1FAAHPARP10PTGES
SCHEMBL7558282 0.83 FFAR1 (0.55) F10FFAR1FAAHTNKSPARP15
SCHEMBL15154989 0.80 F10 (0.45) F10BRS3
SCHEMBL100121 0.79 LOXL2 (0.52) F10LMNASMN1; SMN2
SCHEMBL8599783 0.79 SIRT2 (0.49) F10FFAR1FAAHTNKSPARP15
SCHEMBL8520118 0.77 F10 (0.46) F10FFAR1FAAHTNKSPARP15
SCHEMBL6204785 0.76 TAAR1 (0.57) SMN1; SMN2
SCHEMBL1326762 0.76 CTBP2 (0.60) HTTMMP13SMN1; SMN2
SCHEMBL16301337 0.76 ALDH1A1 (0.45) LMNAHTTSMN1; SMN2
SCHEMBL6754441 0.74 NR1H3 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006033844-A9 4-ARYLSPIROCYCLOALKYL-2-AMINOPYRIMIDINE CARBOXAMIDE KCNQ POTASSIUM CHANNEL MODULATORS BRISTOL MYERS SQUIBB CO (US) 2007-10-25 WO disclosed