SCHEMBL5283360

SCHEMBL5283360

CC(C)(C)OC(=O)N[C@H](CCCOc1cccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)OCC[Si](C)(C)C)c1)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.50
ITGA2B P08514 11/20 0.50
PTPN1 P18031 2/20 0.46
MAPT P10636 2/20 0.45
KLK7 P49862 1/20 0.45
KLK5 Q9Y337 1/20 0.45
ACE P12821 1/20 0.44
PRSS1 P07477 2/20 0.44
PRSS2 P07478 2/20 0.44
PRSS3 P35030 2/20 0.44
TPSAB1 Q15661 2/20 0.44
CTSB P07858 1/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
POLB P06746 1/20 0.43
MAPK1 P28482 1/20 0.43
ITGAV P06756 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5280438 1.00 ITGB3 (0.50) ITGB3ITGA2BPTPN1MAPTKLK7
SCHEMBL5284681 0.96 ITGB3 (0.49) ITGB3ITGA2BPTPN1MAPTACE
SCHEMBL8070826 0.89 ACE (0.53) ITGB3ITGA2BPTPN1MAPTKLK5
SCHEMBL5284506 0.81 ITGB3 (0.46) ITGB3ITGA2BACECTSBCTSS
SCHEMBL4889692 0.81 CTSB (0.47) ITGB3ITGA2BPTPN1ACECTSB
SCHEMBL7709696 0.81 PTPN1 (0.55) PTPN1KLK5ACECTSBCTSS
SCHEMBL20905733 0.81 PTPN1 (0.55) PTPN1KLK5ACECTSBCTSS
SCHEMBL13479127 0.79 CTSS (0.49) ITGB3MAPTKLK7CTSBCTSS
SCHEMBL17773023 0.79 MAPT (0.66) ITGB3ITGA2BMAPTKLK7KLK5
SCHEMBL2552297 0.79 PTPN1 (0.64) ITGB3ITGA2BPTPN1ACECTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007001406-A2 ARYL-CONTAINING MACROCYCLIC COMPOUNDS CHIRON CORPORATION (US) 2007-01-04 WO disclosed