SCHEMBL8070826

SCHEMBL8070826

CC(C)(C)OC(=O)N[C@@H](Cc1cccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)O)c1)C(=O)OCC[Si](C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.53
ITGB3 P05106 7/20 0.50
CTSS P25774 6/20 0.50
ITGA2B P08514 6/20 0.50
CTSK P43235 5/20 0.50
CTSB P07858 4/20 0.50
SYK P43405 1/20 0.49
PPARA Q07869 1/20 0.49
ITGAV P06756 1/20 0.49
CTSL P07711 3/20 0.48
PTPN1 P18031 1/20 0.47
MAPT P10636 1/20 0.47
KLK5 Q9Y337 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5284681 0.90 ITGB3 (0.49) ACEITGB3CTSSITGA2BCTSK
SCHEMBL5280438 0.89 ITGB3 (0.50) ACEITGB3CTSSITGA2BCTSK
SCHEMBL5283360 0.89 ITGB3 (0.50) ACEITGB3CTSSITGA2BCTSK
SCHEMBL4889692 0.88 CTSB (0.47) ACEITGB3CTSSITGA2BCTSK
SCHEMBL8072127 0.87 ACE (0.60) ACEITGB3CTSSITGA2BCTSK
SCHEMBL8072132 0.87 ACE (0.60) ACEITGB3CTSSITGA2BCTSK
SCHEMBL29466819 0.85 CTSL (0.61) CTSSCTSKCTSBCTSL
SCHEMBL10054782 0.84 ACE (0.59) ACEITGB3CTSSITGA2BCTSK
SCHEMBL10054705 0.84 ACE (0.59) ACEITGB3CTSSITGA2BCTSK
SCHEMBL9718080 0.84 SYK (0.57) ITGB3CTSSITGA2BCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080838-A SYNTHETIC CONSTRUCT PREPARED TO HOLD TWO PEPTIDE HELICES IN TIGHT ARRANGEMENT TO MIMIC DNA BINDING CONFORMATION; FOR INVESSTIGATIONAL STUDIES UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2000-06-27 US disclosed