SCHEMBL5285282

SCHEMBL5285282

CCCCCN(C(=O)OCc1ccccc1)c1cc(C(=O)O)cc([N+](=O)[O-])c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.41
ATM Q13315 1/20 0.39
ALDH1A1 P00352 6/20 0.38
PKM P14618 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
RAB9A P51151 3/20 0.37
MAPT P10636 2/20 0.37
AR P10275 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
PDE1C Q14123 1/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4874436 0.82 CCR5 (0.41) ALOX5ATMALDH1A1KMT2ARAB9A
SCHEMBL5346410 0.81 NNMT (0.42) ALDH1A1MAPK1KMT2ATDP1RAB9A
SCHEMBL4868910 0.74 ALDH1A1 (0.48) ALOX5ALDH1A1KMT2ARAB9AMAPT
SCHEMBL11070772 0.73 PAX8 (0.50) ALOX5ALDH1A1MAPK1TDP1RAB9A
SCHEMBL8561986 0.73 KMT2A (0.55) ALOX5ALDH1A1PKMKMT2ATDP1
SCHEMBL5275571 0.73 NOTUM (0.42) ALDH1A1MAPK1TDP1RAB9AMAPT
SCHEMBL2528439 0.73 ALDH1A1 (0.40) ALOX5ALDH1A1KMT2ATDP1RAB9A
SCHEMBL29280745 0.72 ALDH1A1 (0.62) ATMALDH1A1KMT2ATDP1RAB9A
SCHEMBL9299317 0.70 ALDH1A1 (0.51) ATMALDH1A1PKMKMT2ARAB9A
SCHEMBL3938149 0.70 ALDH1A1 (0.37) ALDH1A1KMT2ATDP1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1851208-A1 MACROCYCLIC COMPOUNDS USEFUL AS BACE INHIBITORS Novartis AG (CH) 2007-11-07 EP disclosed
WO-2006074950-A1 MACROCYCLIC COMPOUNDS USEFUL AS BACE INHIBITORS NOVARTIS AG (CH) 2006-07-20 WO disclosed