Morpholine

Morpholine

SCHEMBL5306223

C1COCCN1.CCCNC(=O)c1ccc(-c2ccoc2-c2ccc(C(=O)NCCC)cc2)cc1

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.43
CHRNA10 Q9GZZ6 1/20 0.41
CHRNA9 Q9UGM1 1/20 0.41
GALR1 P47211 1/20 0.39
CD274 Q9NZQ7 6/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
RIPK1 Q13546 1/20 0.38
NAMPT P43490 1/20 0.37
CYP2D6 P10635 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
KCNH2 Q12809 1/20 0.37
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylamine SCHEMBL7878195 0.85 MAPK14 (0.46) MAPK14CHRNA10CHRNA9GALR1HPGD
Morpholine SCHEMBL548401 0.80 MAPK14 (0.44) MAPK14CHRNA10CHRNA9GALR1CD274
Morpholine SCHEMBL5963675 0.79 MAPK14 (0.43) MAPK14CHRNA10CHRNA9GALR1CD274
Dimethylamine SCHEMBL4448304 0.76 MAPK14 (0.44) MAPK14HPGDKMT2ARIPK1CYP2D6
Morpholine SCHEMBL5483585 0.76 OPRD1 (0.41) MAPK14CHRNA10CHRNA9GALR1CD274
SCHEMBL13918749 0.68 KDM4E (0.70) CHRNA10CHRNA9KMT2AKDM4EDRD2
Morpholine SCHEMBL28644462 0.68 LMNA (0.52) CD274HPGDKMT2AKDM4EOPRD1
SCHEMBL1928092 0.65 L3MBTL1 (0.68) MAPK14KMT2AKDM4EDRD2DRD4
SCHEMBL1927649 0.65 DRD2 (0.77) HPGDKMT2AKDM4EDRD2DRD4
SCHEMBL1926646 0.64 HIF1A (0.56) MAPK14HPGDKMT2AKDM4EDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007041677-A9 SOFT TISSUE IMPLANTS AND DRUG COMBINATION COMPOSITIONS, AND USE THEREOF COMBINATORX INC (US) 2007-05-31 WO disclosed
WO-2007041677-A2 SOFT TISSUE IMPLANTS AND DRUG COMBINATION COMPOSITIONS, AND USE THEREOF COMBINATORX, INCORPORATED (US) 2007-04-12 WO disclosed