SCHEMBL5310455

SCHEMBL5310455

O=C(N[C@]1(Cc2ccccc2)CCNC1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.47
ADRB2 P07550 1/20 0.42
USP2 O75604 4/20 0.42
RHOC P08134 1/20 0.40
RHOA P61586 1/20 0.40
SLC6A9 P48067 1/20 0.40
P2RX1 P51575 1/20 0.40
SLC6A4 P31645 6/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A3 Q01959 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP1A2 P05177 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5258355 0.73 ADRB2 (0.39) ADRB2SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL1035119 0.72 PPIA (0.42) ADRB2SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL6122137 0.71 NAMPT (0.57)
SCHEMBL7972011 0.70 SLC6A2 (0.37) ADRB2SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL8824360 0.70 TACR1 (0.63) TACR1SLC6A4
Hydrochloric Acid SCHEMBL9391402 0.70 TACR1 (0.61) TACR1SLC6A4
SCHEMBL6180854 0.70 CHRM3 (0.47)
SCHEMBL9189915 0.69 TACR1 (0.58) TACR1SLC6A4
SCHEMBL5168846 0.68 GRM2 (0.37) ADRB2SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL743634 0.68 CCR2 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007053495-A2 COMPOUNDS USEFUL AS ANTAGONISTS OF CCR2 MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-05-10 WO disclosed