SCHEMBL5314044

SCHEMBL5314044

N#Cc1ccccc1N1C=CC=CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.34
DRD4 P21917 4/20 0.33
DRD2 P14416 3/20 0.33
GRM5 P41594 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HIF1A Q16665 1/20 0.33
NOTUM Q6P988 1/20 0.33
AR P10275 1/20 0.33
GRM1 Q13255 2/20 0.32
KMT2A Q03164 1/20 0.32
RPS6KB1 P23443 1/20 0.32
ROCK1 Q13464 1/20 0.32
DRD3 P35462 2/20 0.31
GRM2 Q14416 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30936310 0.75 DRD4 (0.45) KDM4ETSHRDRD4DRD2GRM5
SCHEMBL29995016 0.74 GRM1 (0.36) GRM1
SCHEMBL29995220 0.74 KDM4E (0.42) KDM4EMAPTDRD4DRD2GRM5
SCHEMBL24163505 0.74 KDM4E (0.38) KDM4ETSHRDRD4DRD2GRM5
SCHEMBL27860451 0.73 KDM4E (0.39) KDM4EMAPTTSHRDRD4DRD2
SCHEMBL7789812 0.73 ALDH1A1 (0.41) KDM4EMAPTTSHRSMN1; SMN2KMT2A
SCHEMBL29958355 0.73
SCHEMBL1238592 0.73 MGLL (0.37)
SCHEMBL9276285 0.73 MGLL (0.37)
SCHEMBL9276325 0.73 KEAP1 (0.41) KDM4EMAPTSMN1; SMN2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869039-A2 PROCESS FOR PREPARING BICYCLIC COMPOUNDS SB Pharmco Puerto Rico Inc. (PR) 2007-12-26 EP claimed
WO-2006108689-A2 PROCESS FOR PREPARING BICYCLIC COMPOUNDS SB PHARMCO PUERTO RICO INC (US) 2006-10-19 WO claimed
EP-3083573-B1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME LLC (US) 2024-08-07 EP disclosed