SCHEMBL5317092

SCHEMBL5317092

[CH2]C(=O)N(C)c1ccc(C#N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.49
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CHRNA4 P43681 1/20 0.49
PGR P06401 4/20 0.46
KMT2A Q03164 1/20 0.46
CA2 P00918 3/20 0.42
CA1 P00915 2/20 0.42
RORC P51449 1/20 0.41
PDK2 Q15119 1/20 0.41
GPBAR1 Q8TDU6 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP2A6 P11509 1/20 0.40
CA12 O43570 1/20 0.40
CA3 P07451 1/20 0.40
CA6 P23280 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7873808 0.82 PGR (0.61) CHRNB2CHRNB4CHRNA3CHRNA4PGR
SCHEMBL9956677 0.81 PGR (0.49) CHRNB2CHRNB4CHRNA3CHRNA4PGR
SCHEMBL10194676 0.80 CCNK (0.47) CHRNB2CHRNB4CHRNA3CHRNA4PGR
SCHEMBL30204212 0.78 ROCK2 (0.48) CHRNB2CHRNB4CHRNA3CHRNA4PGR
SCHEMBL2578635 0.78 CHRNB2 (0.47) CHRNB2CHRNB4CHRNA3CHRNA4PGR
SCHEMBL6170106 0.78 KMT2A (0.54) CHRNB2CHRNB4CHRNA3CHRNA4PGR
SCHEMBL22312043 0.77 KMT2A (0.52) CHRNB2CHRNB4CHRNA3CHRNA4PGR
SCHEMBL6631039 0.75 ALDH1A1 (0.55) KMT2AALDH1A1LMNAMAPTTSHR
SCHEMBL9263725 0.75 APP (0.42) KMT2ACA2CA1PDK2ALDH1A1
Hydrochloric Acid SCHEMBL29472307 0.75 KMT2A (0.51) CHRNB2CHRNB4CHRNA3CHRNA4PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO claimed
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO disclosed