SCHEMBL5318072

SCHEMBL5318072

C[As](C)CCn1c(=O)c2c3cc(OCCO)ccc3c3[nH]c4ccccc4oc3c2c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.37
SIGMAR1 Q99720 2/20 0.33
PPARG P37231 2/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33
NCOA2 Q15596 1/20 0.33
NCOA1 Q15788 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
XDH P47989 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
BCHE P06276 9/20 0.32
ACHE P22303 6/20 0.32
LMNA P02545 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
NR2E3 Q9Y5X4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226141 0.89 SIGMAR1 (0.39) MAOASIGMAR1BCHEACHE
SCHEMBL5228985 0.78 MAOA (0.35) MAOASIGMAR1BCHEACHE
SCHEMBL5226351 0.73 MPO (0.40)
Hydrochloric Acid SCHEMBL5412040 0.72 MPO (0.40) XDH
SCHEMBL5230537 0.71 MPO (0.42) KMT2AMEN1XDHSMN1; SMN2
SCHEMBL5421563 0.69 SIGMAR1 (0.38) SIGMAR1KMT2AL3MBTL1KDR
SCHEMBL5229259 0.66 NR1H2 (0.43) SIGMAR1KMT2AL3MBTL1KDR
SCHEMBL5333498 0.64 MPO (0.44) SIGMAR1KMT2AMEN1XDHSMN1; SMN2
SCHEMBL5231971 0.64 ALDH1A1 (0.34) SIGMAR1PPARGKMT2ARAB9ASMN1; SMN2
SCHEMBL5334632 0.61 CDK4 (0.44) MAOARAB9AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1556387-B1 SUBSTITUTED BENZOL E| 1,4| OXAZINO 3,2-G| ISOINDOLE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2007-04-04 EP claimed