SCHEMBL5319644

SCHEMBL5319644

CC(C)Cn1c(-c2cccc(F)c2F)c(Cl)nc(I)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.36
KDM4E B2RXH2 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GNRHR P30968 2/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
ALDH1A1 P00352 3/20 0.35
TSHR P16473 2/20 0.34
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TRPA1 O75762 1/20 0.34
LMNA P02545 2/20 0.33
THRB P10828 1/20 0.33
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
DYRK1A Q13627 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA1 P30542 1/20 0.32
MDM2 Q00987 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4484784 0.87 SMN1; SMN2 (0.37) TDP1KDM4EAPOBEC3GNPSR1GNRHR
SCHEMBL3986121 0.75 SMN1; SMN2 (0.39) TDP1KDM4EAPOBEC3GNPSR1GNRHR
SCHEMBL3913556 0.70 ALDH1A1 (0.40) TDP1NPSR1GNRHRSMN1; SMN2ALDH1A1
SCHEMBL3985349 0.68 ALDH1A1 (0.34) TDP1NPSR1GNRHRSMN1; SMN2ALDH1A1
SCHEMBL4488011 0.68 SHMT2 (0.38) SMN1; SMN2ALDH1A1L3MBTL1LMNATHRB
SCHEMBL4493753 0.68 CASR (0.38) TDP1NPSR1GNRHRSMN1; SMN2ALDH1A1
SCHEMBL3986025 0.66 HCRTR1 (0.37) NPSR1GNRHRSMN1; SMN2ALDH1A1MEN1
SCHEMBL4483063 0.65 SYK (0.36) TDP1KDM4ENPSR1SMN1; SMN2ALDH1A1
SCHEMBL3991579 0.65 SMN1; SMN2 (0.39) TDP1KDM4EAPOBEC3GNPSR1GNRHR
SCHEMBL4418581 0.64 ADORA2B (0.32) GNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848711-A1 FUNGICIDAL PYRAZINE DERIVATIVES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2007-10-31 EP disclosed
WO-2006089060-A1 FUNGICIDAL PYRAZINE DERIVATIVES E.I. DUPONT DE NEMOURS AND COMPANY (US) 2006-08-24 WO disclosed