SCHEMBL5320802

SCHEMBL5320802

Nc1ccc2c(c1)c(Cc1ccccc1)cn2Cc1ccc(C(F)(F)P(=O)(O)O)c(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
PTPN1 P18031 4/20 0.43
PTPN2 P17706 2/20 0.43
PTPRC P08575 1/20 0.43
PLA2G2A P14555 5/20 0.42
ICMT O60725 9/20 0.42
PLA2G4A P47712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5317466 0.90 HDAC1 (0.45) HDAC1HDAC8HDAC6PTPN1PTPN2
SCHEMBL5342941 0.90 PLA2G2A (0.51) HDAC1HDAC8HDAC6PTPN1PTPN2
SCHEMBL5337560 0.89 HDAC6 (0.55) HDAC1HDAC8HDAC6PTPN1PTPN2
SCHEMBL5320495 0.89 CACNB4 (0.45) HDAC1HDAC8HDAC6PTPN1PTPN2
SCHEMBL5324927 0.89 HDAC1 (0.46) HDAC1HDAC8HDAC6PTPN1PTPN2
SCHEMBL5339333 0.86 PLA2G2A (0.54) HDAC1HDAC8HDAC6PTPN1PTPN2
SCHEMBL5343124 0.77 PTPN1 (0.47) PTPN1PTPN2PTPRC
SCHEMBL5348172 0.76 HDAC6 (0.48) HDAC1HDAC8HDAC6
SCHEMBL5348177 0.76 HDAC6 (0.46) HDAC1HDAC8HDAC6PTPN1PTPN2
SCHEMBL5320081 0.76 PTPN2 (0.45) HDAC1HDAC8HDAC6PTPN1PTPN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007081755-A2 INDOLE-BENZIMIDAZOLE AND INDAZOLE INHIBITORS OF TYROSINE PHOSPHATASES METABASIS THERAPEUTICS, INC. (US) 2007-07-19 WO claimed