SCHEMBL5348172

SCHEMBL5348172

CCOP(=O)(OCC)C(F)(F)c1ccc(Cn2cc(Cc3ccccc3)c3ccccc32)cc1Br

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.48
HDAC1 Q13547 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HTR6 P50406 5/20 0.40
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
CHRNB2 P17787 3/20 0.38
CHRNA7 P36544 3/20 0.38
CHRNA4 P43681 3/20 0.38
HDAC10 Q969S8 3/20 0.38
HDAC3 O15379 2/20 0.37
KMT2A Q03164 1/20 0.37
CYP19A1 P11511 1/20 0.37
HDAC2 Q92769 1/20 0.37
NCOR2 Q9Y618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5337560 0.85 HDAC6 (0.55) HDAC6HDAC1HDAC8HTR6ALDH1A1
SCHEMBL5348177 0.83 HDAC6 (0.46) HDAC6HDAC1HDAC8HTR6ALDH1A1
SCHEMBL5320495 0.78 CACNB4 (0.45) HDAC6HDAC1HDAC8
SCHEMBL5339333 0.78 PLA2G2A (0.54) HDAC6HDAC1HDAC8HTR6ALDH1A1
SCHEMBL5320908 0.77 HTT (0.48) HDAC6HDAC1ALDH1A1LMNA
SCHEMBL5342941 0.77 PLA2G2A (0.51) HDAC6HDAC1HDAC8CHRNB2CHRNA7
SCHEMBL5317466 0.77 HDAC1 (0.45) HDAC6HDAC1HDAC8ALDH1A1LMNA
SCHEMBL5320802 0.76 HDAC1 (0.44) HDAC6HDAC1HDAC8
SCHEMBL5324927 0.76 HDAC1 (0.46) HDAC6HDAC1HDAC8HTR6
SCHEMBL5320081 0.76 PTPN2 (0.45) HDAC6HDAC1HDAC8HTR6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007081755-A2 INDOLE-BENZIMIDAZOLE AND INDAZOLE INHIBITORS OF TYROSINE PHOSPHATASES METABASIS THERAPEUTICS, INC. (US) 2007-07-19 WO disclosed