SCHEMBL5322191

SCHEMBL5322191

CCN1CCC2(CCc3cc(C(=O)NCc4sccc4C)ccc3O2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.42
DRD2 P14416 3/20 0.42
HTR2C P28335 3/20 0.42
RAB9A P51151 2/20 0.39
METAP2 P50579 1/20 0.38
CHRM3 P20309 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
MAOA P21397 1/20 0.37
EPHX2 P34913 2/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14435114 0.79 HTR2A (0.43) HTR2ADRD2HTR2CRAB9ACHRM3
SCHEMBL14435512 0.78 HTR2A (0.48) HTR2ADRD2HTR2CHDAC3HDAC4
SCHEMBL5322616 0.77 RXRA (0.51) HTR2ADRD2HTR2CHDAC3HDAC4
SCHEMBL14435510 0.74 HTR2A (0.42) HTR2ADRD2HTR2CRAB9AHDAC3
SCHEMBL14435508 0.72 EPHX2 (0.48) HTR2ADRD2HTR2CHDAC3HDAC4
SCHEMBL14435509 0.72 TAS1R3 (0.42) HTR2ADRD2HTR2CHDAC3HDAC4
SCHEMBL5325795 0.70 HTR2A (0.44) HTR2ADRD2HTR2CHDAC3HDAC4
SCHEMBL14435119 0.69 NPC1 (0.48) HTR2ADRD2HTR2CRAB9AEPHX2
SCHEMBL14435513 0.68 HTR2A (0.40) HTR2ADRD2HTR2CHDAC3HDAC4
SCHEMBL5320036 0.67 SIGMAR1 (0.46) HTR2ADRD2HTR2CHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007088462-A1 SPIROCHROMANE ANTAGONISTS OF THE H-3 RECEPTOR PFIZER PRODUCTS INC. (US) 2007-08-09 WO disclosed
WO-2007088462-A1 SPIROCHROMANE ANTAGONISTS OF THE H-3 RECEPTOR PFIZER PRODUCTS INC. (US) 2007-08-09 WO disclosed