SCHEMBL5328343

SCHEMBL5328343

O=C1NN=C(C2CCCCC2)c2ccccc2N1Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 7/20 0.48
ALDH1A1 P00352 4/20 0.45
ALDH2 P05091 1/20 0.45
CHRM1 P11229 1/20 0.45
CES1 P23141 1/20 0.45
ALDH3A1 P30838 1/20 0.45
MAPT P10636 2/20 0.40
PKM P14618 1/20 0.40
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
CCKBR P32239 1/20 0.40
TRPA1 O75762 1/20 0.40
CYP19A1 P11511 1/20 0.40
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5328133 0.81 OPRL1 (0.49) PTH1R
SCHEMBL5320618 0.71 PTH1R (0.55) PTH1RALDH1A1MAPTCCKBRAPP
SCHEMBL5320962 0.69 PTH1R (0.56) PTH1RALDH1A1CCKBRHTT
SCHEMBL5280948 0.69 PTH1R (0.76) PTH1RCCKBR
SCHEMBL5323011 0.69 SCN2A (0.46) PTH1RALDH1A1MAPTMEN1KMT2A
SCHEMBL5323577 0.69 PTH1R (0.47) PTH1RALDH1A1MAPTLMNACCKBR
SCHEMBL5287497 0.68 PTH1R (0.50) PTH1RALDH1A1KDM4EMEN1LMNA
SCHEMBL5323683 0.68 PTH1R (0.74) PTH1RCCKBR
SCHEMBL21666455 0.67 ALDH1A1 (0.63) ALDH1A1ALDH2CHRM1CES1ALDH3A1
SCHEMBL2687501 0.66 CCKBR (0.47) CCKBRTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed