SCHEMBL5328133

SCHEMBL5328133

O=C1NN=C(C2CCCCC2)c2ccccc2N1C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 4/20 0.49
OPRM1 P35372 3/20 0.49
OPRK1 P41145 2/20 0.49
CHRM3 P20309 4/20 0.45
CHRM2 P08172 3/20 0.43
ACHE P22303 2/20 0.42
PTH1R Q03431 1/20 0.41
DRD2 P14416 3/20 0.41
DRD4 P21917 3/20 0.41
DRD3 P35462 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5328343 0.81 PTH1R (0.48) PTH1R
SCHEMBL7902547 0.74 OPRL1 (0.56) OPRL1OPRM1OPRK1CHRM3CHRM2
SCHEMBL15847630 0.74 DRD2 (0.68) OPRL1OPRM1OPRK1CHRM3ACHE
SCHEMBL5324889 0.73 OPRL1 (0.46) OPRL1OPRM1OPRK1CHRM3CHRM2
SCHEMBL250673 0.71 ACHE (0.69) OPRL1OPRM1OPRK1CHRM3ACHE
SCHEMBL7447387 0.69 OPRL1 (0.69) OPRL1OPRM1OPRK1CHRM3CHRM2
SCHEMBL1861204 0.69 OPRM1 (0.55) OPRL1OPRM1OPRK1CHRM3ACHE
SCHEMBL1861203 0.69 OPRM1 (0.55) OPRL1OPRM1OPRK1CHRM3ACHE
SCHEMBL13016528 0.68 ACHE (0.67) OPRL1OPRM1OPRK1CHRM3CHRM2
SCHEMBL3075361 0.67 OPRL1 (0.66) OPRL1OPRM1OPRK1CHRM3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed