SCHEMBL5329403

SCHEMBL5329403

CC(C)Oc1ccccc1N1CCN(CCNC(=O)CN2C(=O)C3CC=CCC3C2=O)CC1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 12/20 0.65
ADRA1B P35368 9/20 0.65
ADRA1D P25100 9/20 0.65
HTR1A P08908 1/20 0.48
DRD3 P35462 1/20 0.48
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5302822 0.91 ADRA1A (0.65) ADRA1AADRA1BADRA1DHTR1ADRD3
SCHEMBL5325863 0.90 DRD2 (0.59) ADRA1AADRA1BADRA1DHTR1ADRD3
SCHEMBL5328407 0.88 SLC6A4 (0.55) ADRA1AADRA1BADRA1DHTR1ADRD3
SCHEMBL4530003 0.85 ADRA1A (0.57) ADRA1AADRA1BADRA1DHTR1A
SCHEMBL5306802 0.85 ADRA1A (0.49) ADRA1AADRA1BADRA1DDRD3DRD2
Hydrochloric Acid SCHEMBL4534626 0.84 ADRA1A (0.56) ADRA1AADRA1BADRA1DHTR1A
SCHEMBL5808003 0.83 ADRA1A (0.53) ADRA1AADRA1BADRA1DHTR1ADRD4
SCHEMBL4874588 0.83 ADRA1A (0.56) ADRA1AADRA1BADRA1DHTR1ADRD3
SCHEMBL5423788 0.83 HTR1A (0.57) ADRA1AADRA1BADRA1DHTR1ADRD3
Hydrochloric Acid SCHEMBL5807427 0.82 ADRA1A (0.52) ADRA1AADRA1BADRA1DHTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007029156-A2 ISOINDOLEDIONE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-03-15 WO claimed
WO-2007029156-A2 ISOINDOLEDIONE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-03-15 WO disclosed