SCHEMBL5306802

SCHEMBL5306802

O=C(CN1C(=O)C2CC=CCC2C1=O)NCCN1CCN(c2ccccc2OC2CCCC2)CC1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 5/20 0.49
ADRA1D P25100 4/20 0.49
ADRA1B P35368 4/20 0.49
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5310370 0.90 ADRA1A (0.50) ADRA1AADRA1DADRA1BDRD2DRD3
SCHEMBL5325863 0.87 DRD2 (0.59) ADRA1AADRA1DADRA1BDRD2DRD3
SCHEMBL5328407 0.85 SLC6A4 (0.55) ADRA1AADRA1DADRA1BDRD2DRD3
SCHEMBL4520493 0.85 RAB9A (0.51) ADRA1AADRA1DADRA1BRAB9A
SCHEMBL5329403 0.85 ADRA1A (0.65) ADRA1AADRA1DADRA1BDRD2DRD3
SCHEMBL5310907 0.84 RAB9A (0.46) DRD2DRD3RAB9A
SCHEMBL6213257 0.83 HTR1A (0.54) ADRA1AADRA1DADRA1BDRD2DRD3
Hydrochloric Acid SCHEMBL6215943 0.82 HTR1A (0.53) ADRA1AADRA1DADRA1BDRD2DRD3
SCHEMBL5810923 0.78 RAB9A (0.42) DRD2DRD3RAB9A
SCHEMBL5308285 0.77 DRD2 (0.58) ADRA1AADRA1DADRA1BDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007029156-A2 ISOINDOLEDIONE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-03-15 WO claimed
WO-2007029156-A2 ISOINDOLEDIONE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-03-15 WO disclosed