SCHEMBL5334182

SCHEMBL5334182

CCOC(=O)CSc1nnc(Cc2ccccc2)n1-c1ccccc1

nearest known ligand 0.89

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.89
CYP1A2 P05177 1/20 0.82
CYP3A4 P08684 1/20 0.82
CYP2D6 P10635 1/20 0.82
CYP2C9 P11712 1/20 0.82
CYP2C19 P33261 1/20 0.82
L3MBTL1 Q9Y468 2/20 0.72
ALDH1A1 P00352 8/20 0.72
NPSR1 Q6W5P4 2/20 0.69
MEN1 O00255 3/20 0.65
KMT2A Q03164 3/20 0.65
TSHR P16473 5/20 0.62
HPGD P15428 3/20 0.62
USP2 O75604 2/20 0.62
HSD17B10 Q99714 1/20 0.62
GAA P10253 2/20 0.57
KDM4E B2RXH2 1/20 0.56
MAPT P10636 1/20 0.56
HTT P42858 1/20 0.56
CDC25A P30304 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5332328 0.84 PKM (0.66) PKMCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5331484 0.80 ALDH1A1 (0.66) PKMCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5333083 0.79 MAPT (0.68) PKMCYP3A4CYP2C19L3MBTL1ALDH1A1
SCHEMBL5333033 0.79 ALDH1A1 (0.75) PKML3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL5332243 0.78 ALDH1A1 (0.67) PKML3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL14478938 0.77 ALDH1A1 (0.66) PKMCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5331550 0.76 ALDH1A1 (1.00) PKMCYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL6408488 0.76 ALDH1A1 (0.70) PKML3MBTL1ALDH1A1NPSR1MEN1
SCHEMBL6407843 0.76 NPC1 (0.63) PKMCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL18556577 0.76 POLB (0.73) L3MBTL1ALDH1A1MEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed