SCHEMBL5332328

SCHEMBL5332328

CCOC(=O)CSc1nnc(Cc2ccc3c(c2)OCO3)n1-c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.66
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
CYP2D6 P10635 1/20 0.64
CYP2C9 P11712 1/20 0.64
CYP2C19 P33261 1/20 0.64
POLB P06746 2/20 0.59
ALDH1A1 P00352 9/20 0.54
NPSR1 Q6W5P4 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
RECQL P46063 1/20 0.54
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
TSHR P16473 3/20 0.54
HPGD P15428 2/20 0.53
USP2 O75604 1/20 0.53
MAPK1 P28482 2/20 0.53
HSD17B10 Q99714 1/20 0.51
NPC1 O15118 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5334182 0.84 PKM (0.89) PKMCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5332021 0.84 SMN1; SMN2 (0.74) POLBALDH1A1L3MBTL1KMT2AMEN1
SCHEMBL5332252 0.83 POLB (0.68) CYP3A4CYP2D6POLBALDH1A1NPSR1
SCHEMBL5331032 0.81 POLB (0.62) CYP3A4CYP2D6POLBALDH1A1NPSR1
SCHEMBL5331037 0.81 POLB (0.62) CYP3A4CYP2D6POLBALDH1A1NPSR1
SCHEMBL5332052 0.76 POLB (0.58) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5332046 0.76 POLB (0.58) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5331937 0.72 ADORA1 (0.47) PKMPOLBALDH1A1KMT2AMEN1
SCHEMBL5331484 0.72 ALDH1A1 (0.66) PKMCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5329752 0.72 SMN1; SMN2 (0.83) POLBALDH1A1KMT2ASMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed