SCHEMBL5338742

SCHEMBL5338742

Cc1c(Cl)cccc1S(=O)(=O)Nc1ccc2c(cnn2C)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.50
CCR4 P51679 4/20 0.49
ACLY P53396 1/20 0.48
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
SLC40A1 Q9NP59 1/20 0.46
EDNRB P24530 2/20 0.46
EDNRA P25101 2/20 0.46
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
ACHE P22303 1/20 0.44
TRPM5 Q9NZQ8 1/20 0.44
GSPT1 P15170 1/20 0.43
DDB1 Q16531 1/20 0.43
CRBN Q96SW2 1/20 0.43
NR1I2 O75469 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13106693 0.90 CCR4 (0.61) CCR4ACLYMEN1KMT2ATRPM5
SCHEMBL13106647 0.90 MEN1 (0.57) CCR4ACLYMEN1KMT2AMAOA
SCHEMBL5350340 0.87 HSD11B1 (0.48) HSD11B1CCR4ACLYMEN1KMT2A
SCHEMBL13106642 0.83 MAPT (0.53) ACLYMEN1KMT2ANR1I2
SCHEMBL13106697 0.81 ACLY (0.55) ACLYMEN1KMT2AMAOAMAOB
SCHEMBL13106713 0.81 HTR6 (0.58) NR1I2
SCHEMBL13106696 0.81 ACLY (0.55) ACLYMAOAMAOBACHE
SCHEMBL31702303 0.81 CCR4 (0.61) CCR4MEN1KMT2A
SCHEMBL616054 0.80 NPC1 (0.53) HSD11B1MEN1KMT2ASLC40A1EDNRB
SCHEMBL13106653 0.79 PKM (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7230020-B2 11β-hydroxysteroid dehydrogenase inhibitors STERIX LIMITED (GB) 2007-06-12 US disclosed
US-7230020-B2 11β-hydroxysteroid dehydrogenase inhibitors STERIX LIMITED (GB) 2007-06-12 US disclosed
US-7230020-B2 11β-hydroxysteroid dehydrogenase inhibitors STERIX LIMITED (GB) 2007-06-12 US disclosed
EP-1675844-A1 PHENYL CARBOXAMIDE AND SULFONAMIDE DERIVATIVES FOR USE AS 11-BETA-HYDROXYSTEROID DEHYDROGENASE Sterix Limited (GB) 2006-07-05 EP disclosed
US-20050227987-A1 11beta-hydroxysteroid dehydrogenase inhibitors STERIX LIMITED (GB) 2005-10-13 US disclosed
WO-2005042513-A1 PHENYL CARBOXAMIDE AND SULFONAMIDE DERIVATIVES FOR USE AS 11-BETA-HYDROXYSTEROID DEHYDROGENASE STERIX LIMITED (GB) 2005-05-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050227987-A1 11beta-hydroxysteroid dehydrogenase inhibitors HSD3B1, HSD3B2, HSD17B3 HSD11B1 6/4885CCR4 1963/4885ACLY 356/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.