SCHEMBL5340259

SCHEMBL5340259

CC(=O)c1ccc(-c2cc(F)ccc2NC(=O)c2cn(C)nc2C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.49
POLB P06746 1/20 0.49
STING1 Q86WV6 1/20 0.45
WDR5 P61964 2/20 0.44
NTRK1 P04629 3/20 0.42
GAA P10253 3/20 0.41
KDM4E B2RXH2 1/20 0.41
NPSR1 Q6W5P4 5/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
HPGD P15428 1/20 0.40
CHRM3 P20309 2/20 0.40
NR3C1 P04150 1/20 0.40
PGR P06401 1/20 0.40
MAPK1 P28482 1/20 0.40
NTRK2 Q16620 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1136137 0.93 LMNA (0.54) LMNAPOLBSTING1WDR5NTRK1
SCHEMBL1136025 0.90 LMNA (0.51) LMNAPOLBSTING1WDR5NTRK1
SCHEMBL1136177 0.89 LMNA (0.64) LMNAPOLBSTING1WDR5NTRK1
SCHEMBL9979648 0.89 LMNA (0.45) LMNAPOLBSTING1WDR5NTRK1
SCHEMBL13491717 0.89 LMNA (0.52) LMNAPOLBWDR5NTRK1GAA
SCHEMBL16618150 0.88 LMNA (0.63) LMNAPOLBWDR5NTRK1NPSR1
SCHEMBL1144935 0.87 LMNA (0.53) LMNAPOLBSTING1WDR5NTRK1
SCHEMBL29445385 0.85 LMNA (0.53) LMNAPOLBSTING1WDR5NTRK1
SCHEMBL29445400 0.85 LMNA (0.48) LMNAPOLBWDR5NTRK1GAA
SCHEMBL303303 0.85 LMNA (0.53) LMNAPOLBSTING1WDR5NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1305292-B1 BIPHENYL CARBOXAMIDES BAYER CROPSCIENCE AG (DE) 2012-06-20 EP disclosed
US-7176228-B2 Pyrazole biphenylcarboxamides BAYER CROPSCIENCE AG (DE) 2007-02-13 US disclosed
US-7176228-B2 Pyrazole biphenylcarboxamides BAYER CROPSCIENCE AG (DE) 2007-02-13 US disclosed
US-7176228-B2 Pyrazole biphenylcarboxamides BAYER CROPSCIENCE AG (DE) 2007-02-13 US disclosed
US-20040039043-A1 Biphenyl carboxamides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2004-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039043-A1 Biphenyl carboxamides CYP1A1, AHR, CYP1B1 LMNA 2098/4885POLB 1251/4885STING1 3038/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.