SCHEMBL5350293

SCHEMBL5350293

O=C(O)c1ccc(CCCc2ccncc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.59
TBXAS1 P24557 2/20 0.58
RARB P10826 6/20 0.56
ALDH1A1 P00352 2/20 0.53
MEN1 O00255 1/20 0.53
RARA P10276 1/20 0.53
MAPT P10636 1/20 0.53
MTOR P42345 1/20 0.53
KMT2A Q03164 1/20 0.53
NAMPT P43490 1/20 0.51
PTGER1 P34995 1/20 0.48
PTGER4 P35408 1/20 0.48
PTGER3 P43115 1/20 0.48
PTGER2 P43116 1/20 0.48
HDAC8 Q9BY41 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10638830 0.96 NAPRT (0.59) NAPRTTBXAS1RARBALDH1A1MEN1
SCHEMBL6769826 0.92 NAPRT (0.64) NAPRTTBXAS1RARBALDH1A1MEN1
Hydrochloric Acid SCHEMBL3896488 0.90 NAPRT (0.61) NAPRTTBXAS1RARBALDH1A1MEN1
SCHEMBL133470 0.88 RARB (0.68) TBXAS1RARBALDH1A1MEN1RARA
SCHEMBL18906031 0.84 HDAC1 (0.65) NAPRTALDH1A1MEN1KMT2ANAMPT
SCHEMBL371605 0.83 RARB (0.71) TBXAS1RARBALDH1A1MEN1RARA
SCHEMBL7405035 0.83 PLA2G4B (0.58) TBXAS1ALDH1A1MEN1KMT2ATP53
SCHEMBL1982703 0.82 HDAC8 (0.67) NAPRTRARBALDH1A1MEN1RARA
SCHEMBL9472454 0.81 RARB (0.72) TBXAS1RARBALDH1A1MEN1RARA
SCHEMBL30053056 0.81 RARB (0.72) TBXAS1RARBALDH1A1MEN1RARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7300934-B2 Benzamide nitriles ROCHE PALO ALTO LLC (US) 2007-11-27 US disclosed
EP-1633701-A1 BENZAMIDE NITRILE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-03-15 EP disclosed
WO-2004106285-A1 BENZAMIDE NITRILE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-12-09 WO disclosed
US-20040248949-A1 Benzamide nitriles ROCHE PALO ALTO LLC 2004-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040248949-A1 Benzamide nitriles CTSK, CTSS, CMA1 NAPRT 1375/4885TBXAS1 1958/4885RARB 2823/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.