SCHEMBL535063

SCHEMBL535063

O=C(O)N1CCC(O)(c2ccc(F)c(F)c2)CC1C#CBr

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.39
CCR2 P41597 1/20 0.35
CCR1 P32246 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL557091 0.74 CCR2 (0.33) DRD2CCR2
SCHEMBL3384526 0.72 DRD2 (0.45) DRD2CCR1
SCHEMBL534534 0.71 OPRD1 (0.36) CCR2
SCHEMBL2531562 0.70 DRD2 (0.41) DRD2CCR2CCR1
SCHEMBL535062 0.68 DRD2 (0.41) DRD2
SCHEMBL2430891 0.67 CCR2 (0.38) DRD2CCR2
SCHEMBL3386011 0.67 KCNN4 (0.39) DRD2
SCHEMBL2534655 0.66 CCR2 (0.40) DRD2CCR2
SCHEMBL16422879 0.65 DRD2 (0.45) DRD2CCR1
SCHEMBL556468 0.65 CCR2 (0.34) DRD2CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed