SCHEMBL534534

SCHEMBL534534

O=C(O)N1CC[C@](O)(c2ccc(F)c(F)c2)[C@@H](C#CBr)C1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 9/20 0.36
OPRK1 P41145 9/20 0.36
OPRM1 P35372 4/20 0.36
CCR2 P41597 1/20 0.33
RORC P51449 1/20 0.33
SLC6A3 Q01959 4/20 0.33
KMT2A Q03164 1/20 0.33
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
MC4R P32245 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL534472 0.88 OPRD1 (0.37) OPRD1OPRK1OPRM1CCR2RORC
SCHEMBL557090 0.84 RORC (0.39) RORC
SCHEMBL557091 0.75 CCR2 (0.33) CCR2RORCSLC6A3KMT2AMC4R
SCHEMBL533858 0.73 REN (0.46)
SCHEMBL3384526 0.73 DRD2 (0.45) OPRD1OPRK1OPRM1KMT2A
SCHEMBL556467 0.73 RORC (0.40) RORC
SCHEMBL16423307 0.71 RORC (0.42) OPRD1OPRK1OPRM1RORCSLC6A3
SCHEMBL16423136 0.71 SLC6A3 (0.41) OPRD1OPRK1OPRM1SLC6A3KMT2A
SCHEMBL535063 0.71 DRD2 (0.39) CCR2
SCHEMBL556661 0.71 RORC (0.40) OPRD1OPRK1OPRM1RORCSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed