SCHEMBL5354451

SCHEMBL5354451

COc1ccc2c(cc(/C=C/C(=O)OC(C)(C)C)n2Cc2ccccc2)c1OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
PTGER4 P35408 2/20 0.40
PTGER2 P43116 2/20 0.40
PTGER3 P43115 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
APP P05067 5/20 0.39
HDAC8 Q9BY41 1/20 0.39
TSHR P16473 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
KMT2A Q03164 1/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
CA12 O43570 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5354456 1.00 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDPTGER4PTGER2
SCHEMBL5362181 0.79 MEN1 (0.42) ALDH1A1KDM4EGAAMAPTPKM
SCHEMBL5362177 0.79 MEN1 (0.42) ALDH1A1KDM4EGAAMAPTPKM
SCHEMBL5369798 0.77 SRD5A2 (0.43) ALDH1A1KDM4EPTGER3PKMHDAC8
SCHEMBL5372569 0.77 SRD5A2 (0.43) ALDH1A1KDM4EPTGER3PKMHDAC8
SCHEMBL5363418 0.76 CCR2 (0.49) ALDH1A1KDM4EHPGDGAAMAPT
SCHEMBL5359096 0.76 CCR2 (0.49) ALDH1A1KDM4EHPGDGAAMAPT
SCHEMBL5427991 0.73 CCR2 (0.43) MAPTMTNR1AMTNR1B
SCHEMBL5427985 0.73 CCR2 (0.43) MAPTMTNR1AMTNR1B
SCHEMBL5350992 0.72 MAPT (0.43) ALDH1A1KDM4EGAAMAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007134421-A1 2-VINYL INDOLES, PYRIDO AND AZEPINO INDOLE DERIVATIVES, 2-ALKYNYL INDOLES, 2-ALKYNYL BENZO[b]FURANS, THEIR PRECURSORS AND NOVEL PROCESSES FOR THE PREPARATION THEREOF LAUTENS MARK (CA) 2007-11-29 WO disclosed