SCHEMBL5355232

SCHEMBL5355232

Cc1cc(C(F)(C(F)(F)F)C(F)(F)F)cc(C)c1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.48
ESR2 Q92731 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
PTGS1 P23219 7/20 0.39
PTGS2 P35354 7/20 0.39
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 1/20 0.37
ALOX5 P09917 6/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GAA P10253 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
ACHE P22303 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL697862 0.89 ESR1 (0.43) ESR1ESR2CA1CA2PTGS1
SCHEMBL22927041 0.81 RAPGEF4 (0.34) MAPTGAA
SCHEMBL247818 0.80 ESR1 (0.48) ESR1ESR2CA1CA2PTGS1
SCHEMBL9861932 0.79 CA1 (0.52) ESR1ESR2CA1CA2PTGS1
SCHEMBL11126670 0.78 ESR1 (0.46) ESR1ESR2CA1CA2PTGS1
SCHEMBL3682450 0.78 ESR1 (0.46) ESR1ESR2CA1CA2PTGS1
SCHEMBL17286709 0.76 ESR1 (0.45) ESR1ESR2CA1CA2PTGS1
SCHEMBL2837831 0.76 ESR1 (0.45) ESR1ESR2CA1CA2PTGS1
SCHEMBL10643173 0.76 ESR1 (0.45) ESR1ESR2CA1CA2PTGS1
SCHEMBL3140759 0.75 AGBL2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169955-B2 Perfluoroisopropylbenzene derivative NIHON NOHYAKU CO., LTD. (JP) 2007-01-30 US disclosed
US-20050113567-A1 Perfluoroisopropylbenzene derivative NIHON NOHYAKU CO., LTD. (JP) 2005-05-26 US disclosed
US-20030187233-A1 PERFLUOROISOPROPYBENZENE DERIVATIVE NIHON NOHYAKU CO., LTD. (JP) 2003-10-02 US disclosed
EP-1253128-A1 PERFLUOROISOPROPYLBENZENE DERIVATIVES Nihon Nohyaku Co., Ltd. (JP) 2002-10-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030187233-A1 PERFLUOROISOPROPYBENZENE DERIVATIVE AFF1, CBR1, RER1 ESR1 1830/4885ESR2 977/4885CA1 3258/4885
US-20050113567-A1 Perfluoroisopropylbenzene derivative FFAR3, CBR3, HCAR3 ESR1 361/4885ESR2 728/4885CA1 2489/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.