SCHEMBL5355906

SCHEMBL5355906

COc1cccc2cc(C=CC(=O)OC(C)(C)C)[nH]c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
HRH4 Q9H3N8 2/20 0.42
FLT3 P36888 2/20 0.42
IDO1 P14902 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
ESR1 P03372 1/20 0.38
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
ITK Q08881 2/20 0.36
GAA P10253 2/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
RECQL P46063 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5355901 1.00 MTNR1A (0.43) MTNR1AMTNR1BHRH4FLT3IDO1
SCHEMBL5360581 0.78 ATP6V1B1 (0.51) FLT3IDO1KDM4EDRD3MAPT
SCHEMBL5360579 0.78 ATP6V1B1 (0.51) FLT3IDO1KDM4EDRD3MAPT
SCHEMBL26611680 0.76 ABCG2 (0.59) KDM4EALDH1A1ESR1MAPTSMN1; SMN2
SCHEMBL24557535 0.76 ABCG2 (0.59) KDM4EALDH1A1ESR1MAPTSMN1; SMN2
SCHEMBL20920169 0.74 ALDH1A1 (0.49) MTNR1AMTNR1BHRH4FLT3IDO1
SCHEMBL19244392 0.72 NFE2L2 (0.66) KDM4EALDH1A1MEN1MAPTHPGD
SCHEMBL19244393 0.72 NFE2L2 (0.66) KDM4EALDH1A1MEN1MAPTHPGD
SCHEMBL20937296 0.71 ITK (0.44) MTNR1AMTNR1BHRH4FLT3IDO1
SCHEMBL30407949 0.71 FLT3 (0.43) HRH4FLT3KDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007134421-A1 2-VINYL INDOLES, PYRIDO AND AZEPINO INDOLE DERIVATIVES, 2-ALKYNYL INDOLES, 2-ALKYNYL BENZO[b]FURANS, THEIR PRECURSORS AND NOVEL PROCESSES FOR THE PREPARATION THEREOF LAUTENS MARK (CA) 2007-11-29 WO disclosed