SCHEMBL536016

SCHEMBL536016

Nc1nc(N)nc(NCc2ncccn2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 3/20 0.49
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
GPR68 Q15743 4/20 0.39
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
HTT P42858 1/20 0.39
HSP90AA1 P07900 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALOX15 P16050 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ADORA2A P29274 2/20 0.38
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL540957 0.78 KCNH3 (0.86) KCNH3SMN1; SMN2KDM4EALDH1A1
SCHEMBL27609444 0.77 MAOA (0.60) NPC1RAB9ASMN1; SMN2HTTKDM4E
SCHEMBL536394 0.75 KCNH3 (0.52) KCNH3GPR68NPC1RAB9ASMN1; SMN2
SCHEMBL3301514 0.71 NPSR1 (0.74) KCNH3CA1CA2CA9NPSR1
SCHEMBL1923771 0.69 KCNH3 (0.82) KCNH3KDM4EGAA
SCHEMBL29167130 0.69 CA1 (0.57) KCNH3CA1CA2CA9NPSR1
Hydrochloric Acid SCHEMBL9247173 0.69 NPSR1 (0.72) KCNH3CA1CA2CA9NPSR1
SCHEMBL380440 0.69 CA1 (0.47) CA1CA2CA9NPSR1GPR68
SCHEMBL5906873 0.69 CA1 (0.42) CA1CA2CA9NPSR1GPR68
SCHEMBL15294300 0.67 CA1 (0.41) CA1CA2CA9NPSR1GPR68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414351-A1 NOVEL SALT OF 1,3,5-TRIAZINE-2,4,6-TRIAMINE DERIVATIVE Astellas Pharma Inc. (JP) 2012-02-08 EP disclosed
WO-2010114162-A1 NOVEL SALT OF 1,3,5-TRIAZINE-2,4,6-TRIAMINE DERIVATIVE ASTELLAS PHARMA INC. (JP) 2010-10-07 WO disclosed