SCHEMBL536394

SCHEMBL536394

Nc1nc(NCc2ncccn2)nc(N(c2ccc(F)cc2)c2ccc(F)cc2)n1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 5/20 0.52
NPC1 O15118 1/20 0.41
JAK2 O60674 1/20 0.41
RAB9A P51151 1/20 0.41
MAPT P10636 2/20 0.39
HTR2C P28335 1/20 0.39
HTR7 P34969 1/20 0.39
APP P05067 1/20 0.37
GPR68 Q15743 2/20 0.36
MAPK1 P28482 1/20 0.36
ADORA2A P29274 2/20 0.35
SCN9A Q15858 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1925175 0.82 KCNH3 (0.51) KCNH3HTR2CHTR7APPGPR68
SCHEMBL540957 0.77 KCNH3 (0.86) KCNH3MAPK1SMN1; SMN2
SCHEMBL536016 0.75 KCNH3 (0.49) KCNH3NPC1RAB9AAPPGPR68
SCHEMBL1280999 0.69 KCNH3 (1.00) KCNH3
SCHEMBL1282106 0.68 ALDH1A1 (0.50) NPC1JAK2RAB9AMAPTADORA2A
SCHEMBL29223873 0.66 CA1 (0.60) KCNH3HTR2CHTR7APPGPR68
SCHEMBL535908 0.66 KCNH3 (1.00) KCNH3
SCHEMBL28451024 0.66 MAPT (0.54) NPC1JAK2RAB9AMAPTHTR7
SCHEMBL15721117 0.64 HTR7 (0.46) KCNH3HTR2CHTR7ADORA2A
SCHEMBL581128 0.63 MAPT (0.54) KCNH3NPC1JAK2RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414351-A1 NOVEL SALT OF 1,3,5-TRIAZINE-2,4,6-TRIAMINE DERIVATIVE Astellas Pharma Inc. (JP) 2012-02-08 EP disclosed
WO-2010114162-A1 NOVEL SALT OF 1,3,5-TRIAZINE-2,4,6-TRIAMINE DERIVATIVE ASTELLAS PHARMA INC. (JP) 2010-10-07 WO disclosed