SCHEMBL536112

SCHEMBL536112

O=C(O)c1cccc2nc(-c3ccc(-c4ccccc4)c(F)c3F)[nH]c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
RAB9A P51151 2/20 0.49
DHODH Q02127 11/20 0.47
POLB P06746 1/20 0.44
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4A O75164 1/20 0.41
KDM5A P29375 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM5B Q9UGL1 1/20 0.41
GPR17 Q13304 1/20 0.41
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPT P10636 1/20 0.40
PIM1 P11309 1/20 0.40
GFER P55789 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL505457 0.84 DHODH (0.68) KDM4ERAB9ADHODHKDM4AKDM5A
SCHEMBL696548 0.83 DHODH (0.56) KDM4ERAB9ADHODHPOLBCYP1A2
SCHEMBL536118 0.83 DHODH (0.52) DHODHCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6840296 0.83 RAB9A (0.56) KDM4ERAB9ADHODHPOLBALDH1A1
SCHEMBL536113 0.82 DHODH (0.58) KDM4ERAB9ADHODHALDH1A1HPGD
SCHEMBL506154 0.81 DHODH (0.67) KDM4ERAB9ADHODH
SCHEMBL505378 0.80 DHODH (0.69) KDM4ERAB9ADHODHALDH1A1NPC1
SCHEMBL536111 0.79 DHODH (0.59) KDM4ERAB9ADHODHALDH1A1NPC1
SCHEMBL6840189 0.79 PIN1 (0.58) KDM4ERAB9ADHODHALDH1A1KDM4A
SCHEMBL6840235 0.79 TNKS (0.54) KDM4ERAB9ADHODHALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414328-A2 DIHYDROOROTATE DEHYDROGENASE INHIBITORS Merck Serono S.A. (CH) 2012-02-08 EP disclosed