SCHEMBL5362192

SCHEMBL5362192

COCCS(=O)(=O)c1nc(C(O)c2ccc(C)cc2)ns1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.33
HPGD P15428 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HTT P42858 1/20 0.33
CYP2C19 P33261 4/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
CYP1A2 P05177 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP3A4 P08684 2/20 0.30
CYP2D6 P10635 1/20 0.30
MAPT P10636 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5359842 0.86 LMNA (0.33) LMNAHPGDALDH1A1HTTCYP2C19
SCHEMBL5362184 0.72 NPC1 (0.40) LMNAHPGDALDH1A1HTTSMN1; SMN2
SCHEMBL5288067 0.68 LOX (0.34)
SCHEMBL5306313 0.68 LOX (0.31)
SCHEMBL5368956 0.66
SCHEMBL5304859 0.66 NAMPT (0.33) HPGDALDH1A1CYP2C19CYP1A2CYP3A4
SCHEMBL564467 0.65 ALDH1A1 (0.64) LMNAHPGDALDH1A1HTTCYP2C19
SCHEMBL5297823 0.64 KMT2A (0.35) LMNAHPGDALDH1A1SMN1; SMN2CYP3A4
SCHEMBL5299127 0.63 ADORA3 (0.32)
SCHEMBL5299398 0.63 KCNH3 (0.44) LMNAALDH1A1SMN1; SMN2MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO claimed
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO disclosed