SCHEMBL5364064

SCHEMBL5364064

CCOC(Cc1ccc(OCc2ccccc2)cc1)C(=O)OC

nearest known ligand 0.73

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 11/20 0.73
PPARG P37231 9/20 0.73
PPARD Q03181 5/20 0.73
LTA4H P09960 2/20 0.62
LMNA P02545 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
ALOX5 P09917 1/20 0.54
ALDH1A1 P00352 1/20 0.52
LAP3 P28838 1/20 0.52
GAA P10253 1/20 0.52
RAB9A P51151 1/20 0.52
FFAR1 O14842 1/20 0.51
FFAR4 Q5NUL3 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7191581 1.00 PPARA (0.73) PPARAPPARGPPARDLTA4HLMNA
SCHEMBL15811673 0.91 PPARA (0.75) PPARAPPARGPPARDLTA4HLMNA
SCHEMBL4758109 0.91 PPARA (0.75) PPARAPPARGPPARDLTA4HLMNA
SCHEMBL5338861 0.91 PPARA (0.75) PPARAPPARGPPARDLTA4HLMNA
Hydrochloric Acid SCHEMBL7212899 0.90 PPARA (0.73) PPARAPPARGPPARDLTA4HLMNA
Hydrochloric Acid SCHEMBL7212895 0.90 PPARA (0.73) PPARAPPARGPPARDLTA4HLMNA
SCHEMBL4758161 0.89 PPARA (0.60) PPARAPPARGPPARDLTA4H
SCHEMBL16415813 0.88 PPARA (0.92) PPARAPPARGPPARD
SCHEMBL5993963 0.88 PPARA (0.92) PPARAPPARGPPARD
SCHEMBL5608022 0.88 PPARA (0.92) PPARAPPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100376560-C New tricyclic compounds and their use in medicine, process for their preparation and pharmaceutical compositions containing them REDDY CHEMINOR INC (IN) 2008-03-26 CN disclosed
US-20070276138-A1 Modulators of peroxisome proliferator activated receptors BROOKS DAWN A 2007-11-29 US disclosed
US-20070276138-A1 Modulators of peroxisome proliferator activated receptors BROOKS DAWN A 2007-11-29 US disclosed
US-20070276138-A1 Modulators of peroxisome proliferator activated receptors BROOKS DAWN A 2007-11-29 US disclosed
US-7220880-B2 Amide linker peroxisome proliferator activated receptor modulators ELI LILLY AND COMPANY (US) 2007-05-22 US disclosed
US-7220880-B2 Amide linker peroxisome proliferator activated receptor modulators ELI LILLY AND COMPANY (US) 2007-05-22 US disclosed
US-7220880-B2 Amide linker peroxisome proliferator activated receptor modulators ELI LILLY AND COMPANY (US) 2007-05-22 US disclosed
US-7192982-B2 Modulators of peroxisome proliferator activated receptors LIGAND PHARMACEUTICALS, INC. (US) 2007-03-20 US disclosed
US-7192982-B2 Modulators of peroxisome proliferator activated receptors LIGAND PHARMACEUTICALS, INC. (US) 2007-03-20 US disclosed
US-7192982-B2 Modulators of peroxisome proliferator activated receptors LIGAND PHARMACEUTICALS, INC. (US) 2007-03-20 US disclosed
US-20020177726-A1 Process for the preparation of 3-aryl-2-hydroxy propanoic acid DR. REDDY'S RESEARCH FOUNDATION 2002-11-28 US disclosed
US-6440961-B1 Tricyclic compounds and their use in medicine: process for their preparation and pharmaceutical compositions containing them DR. REDDY'S RESEARCH FOUNDATION (IN) 2002-08-27 US disclosed
US-20020077320-A1 Novel tricyclic compounds and their use in medicine; process for their preparation and pharmaceutical compositions containing them DR. REDDY'S RESEARCH FOUNDATION AND REDDY- CHEMINOR, INC. 2002-06-20 US disclosed
CN-1352639-A Novel tricyclic compounds and their use in medicine, process for their production and pharmaceutical composition containing them REDDY RESEARCH FOUNDATION (IN) 2002-06-05 CN disclosed
WO-2002024625-A2 PROCESS FOR THE PREPARATION OF 3-ARYL-2-HYDROXY PROPANOIC ACID DERIVATIVES DR. REDDY'S RESEARCH FOUNDATION (IN) 2002-03-28 WO disclosed
EP-1155006-A1 NOVEL TRICYCLIC COMPOUNDS AND THEIR USE IN MEDICINE; PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEM Dr. Reddy's Research Foundation (IN) 2001-11-21 EP disclosed
CN-1280575-A Novel tricyclic compounds and their use as medicaments, process for their preparation and pharmaceutical compositions containing them REDDY CHEMINOR INC (IN) 2001-01-17 CN disclosed
EP-1049684-A1 NOVEL TRICYCLIC COMPOUNDS AND THEIR USE IN MEDICINE; PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-11-08 EP disclosed
WO-2000050414-A1 NOVEL TRICYCLIC COMPOUNDS AND THEIR USE IN MEDICINE; PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEM DR.REDDY'S RESEARCH FOUNDATION (IN) 2000-08-31 WO disclosed
WO-1999019313-A1 NOVEL TRICYCLIC COMPOUNDS AND THEIR USE IN MEDICINE; PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1999-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020077320-A1 Novel tricyclic compounds and their use in medicine; process for their preparation and pharmaceutical compositions containing them LIPC, GPR119, CPT1A PPARA 281/4885PPARG 102/4885PPARD 308/4885
US-20020177726-A1 Process for the preparation of 3-aryl-2-hydroxy propanoic acid HPD, HAO1, HAAO PPARA 265/4885PPARG 772/4885PPARD 581/4885
US-20070276138-A1 Modulators of peroxisome proliferator activated receptors PPARG, NCOA4, PPARA PPARA 3/4885PPARG 1/4885PPARD 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.