SCHEMBL5364790

SCHEMBL5364790

CC(Oc1ccccc1)C(=O)N1CCC(CNC(=O)c2ccc(O)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.54
PKM P14618 1/20 0.54
CHRM4 P08173 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
APOBEC3A P31941 1/20 0.47
APOBEC3G Q9HC16 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
TPSAB1 Q15661 4/20 0.47
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367904 0.81 ME2 (0.56) KDM4EPKMCHRM4MEN1KMT2A
SCHEMBL6536256 0.79 KDM4E (0.55) KDM4EPKMCHRM4MEN1KMT2A
SCHEMBL5368103 0.77 TPSAB1 (0.71) KDM4EPKMCHRM4HDAC3HDAC4
SCHEMBL5368399 0.77 HDAC3 (0.53) KDM4EPKMCHRM4HDAC3HDAC4
SCHEMBL5362915 0.75 HDAC6 (0.60) KDM4EPKMCHRM4HDAC3HDAC4
SCHEMBL5523321 0.75 HDAC3 (0.51) CHRM4MEN1KMT2AHDAC3HDAC4
SCHEMBL5521812 0.75 HDAC3 (0.51) CHRM4MEN1KMT2AHDAC3HDAC4
SCHEMBL5521806 0.75 HDAC3 (0.51) CHRM4MEN1KMT2AHDAC3HDAC4
SCHEMBL2400940 0.74 ITGB3 (0.42) KDM4EPKMMEN1KMT2AAPOBEC3A
SCHEMBL5371009 0.74 PKM (0.51) KDM4EPKMCHRM4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed