SCHEMBL5367569

SCHEMBL5367569

COC(=O)c1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)nc1Cn1c(C)c(C(=O)OC(C)(C)C)c(-c2ccc(C#N)cc2)c1C

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AR P10275 13/20 0.57
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
NTRK1 P04629 1/20 0.32
NTRK2 Q16620 1/20 0.32
PIN1 Q13526 1/20 0.31
SLC34A1 Q06495 1/20 0.31
FNTA P49354 2/20 0.31
FNTB P49356 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5359676 0.91 AR (0.53) ARNTRK1NTRK2FNTAFNTB
SCHEMBL5362447 0.90 AR (0.52) ARNTRK1NTRK2FNTAFNTB
SCHEMBL5365950 0.83 AR (0.44) ARNTRK1NTRK2FNTAFNTB
SCHEMBL5364006 0.75 AR (0.52) ARSLC34A1FNTAFNTB
SCHEMBL5367629 0.74 AR (0.44) AR
SCHEMBL6468911 0.74 AR (1.00) ARALDH1A1LMNA
SCHEMBL5358998 0.72 AR (0.54) ARFNTAFNTB
SCHEMBL5359896 0.72 AR (0.43) ARNTRK1NTRK2SLC34A1FNTA
SCHEMBL6465312 0.71 AR (0.89) ARLMNA
SCHEMBL5361541 0.70 AR (0.51) ARALDH1A1LMNASLC34A1FNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed