SCHEMBL5365950

SCHEMBL5365950

CCc1c(C(=O)OC(C)(C)C)c(-c2ccc(C#N)cc2)c(C)n1Cc1nn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1C

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.44
GRIA2 P42262 3/20 0.34
GRIA4 P48058 3/20 0.34
NTRK1 P04629 1/20 0.33
NTRK2 Q16620 1/20 0.33
FNTA P49354 2/20 0.32
FNTB P49356 2/20 0.32
BRD4 O60885 1/20 0.30
CRHBP P24387 1/20 0.30
CRHR2 Q13324 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5359676 0.92 AR (0.53) ARNTRK1NTRK2FNTAFNTB
SCHEMBL5367629 0.90 AR (0.44) ARGRIA2GRIA4
SCHEMBL5362447 0.85 AR (0.52) ARNTRK1NTRK2FNTAFNTB
SCHEMBL5367569 0.83 AR (0.57) ARNTRK1NTRK2FNTAFNTB
SCHEMBL5359896 0.82 AR (0.43) ARGRIA2GRIA4NTRK1NTRK2
SCHEMBL5360480 0.74 AR (0.42) ARGRIA2GRIA4FNTAFNTB
SCHEMBL5358998 0.70 AR (0.54) ARGRIA2GRIA4FNTAFNTB
SCHEMBL5364006 0.69 AR (0.52) ARFNTAFNTBBRD4
SCHEMBL5358573 0.67 AR (0.54) ARGRIA2GRIA4
SCHEMBL5369671 0.67 AR (0.60) ARGRIA2GRIA4NTRK1NTRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed