SCHEMBL5359896

SCHEMBL5359896

CCc1c(C(=O)OC(C)(C)C)c(-c2ccc(C#N)cc2)c(C)n1Cc1cc(C#N)n(C(c2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.43
NTRK1 P04629 1/20 0.34
NTRK2 Q16620 1/20 0.34
GRIA2 P42262 3/20 0.33
GRIA4 P48058 3/20 0.33
BRD4 O60885 1/20 0.32
FNTA P49354 2/20 0.31
FNTB P49356 2/20 0.31
SLC34A1 Q06495 1/20 0.31
ACSS2 Q9NR19 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5365950 0.82 AR (0.44) ARNTRK1NTRK2GRIA2GRIA4
SCHEMBL5360480 0.79 AR (0.42) ARGRIA2GRIA4BRD4FNTA
SCHEMBL5362447 0.75 AR (0.52) ARNTRK1NTRK2FNTAFNTB
SCHEMBL5359676 0.74 AR (0.53) ARNTRK1NTRK2FNTAFNTB
SCHEMBL5367569 0.72 AR (0.57) ARNTRK1NTRK2FNTAFNTB
SCHEMBL5367629 0.72 AR (0.44) ARGRIA2GRIA4
SCHEMBL5358998 0.69 AR (0.54) ARGRIA2GRIA4BRD4FNTA
SCHEMBL5370036 0.66 AR (0.49) ARBRD4FNTAFNTBSLC34A1
SCHEMBL5369671 0.66 AR (0.60) ARNTRK1NTRK2GRIA2GRIA4
SCHEMBL5361541 0.66 AR (0.51) ARBRD4FNTAFNTBSLC34A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed