SCHEMBL539376

SCHEMBL539376

O=C1CCN(C2(c3ccc(F)cc3)CC2I)CC1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.36
MAOB P27338 2/20 0.36
MAOA P21397 1/20 0.36
DPP4 P27487 2/20 0.33
POLB P06746 1/20 0.32
SLC6A9 P48067 3/20 0.32
OPRM1 P35372 2/20 0.32
KCNH2 Q12809 1/20 0.32
TACR1 P25103 3/20 0.32
ALDH1A1 P00352 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
LIG1 P18858 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL426911 0.73 SLC6A9 (0.45) HSD11B1SLC6A9OPRM1KCNH2GRIN2B
SCHEMBL23780914 0.71 LMNA (0.49) POLBALDH1A1
SCHEMBL11594047 0.65 CCR1 (0.41) HSD11B1OPRM1KCNH2TACR1ALDH1A1
SCHEMBL10676298 0.63 MEN1 (0.63) HSD11B1MAOBMAOAALDH1A1LIG1
SCHEMBL61987 0.63 ALDH1A1 (0.55) POLBALDH1A1
SCHEMBL2761726 0.61 GAA (0.40) ALDH1A1CYP1A2CYP3A4
SCHEMBL11594099 0.61 HSD11B1 (0.33) HSD11B1SLC6A9OPRM1
SCHEMBL5768239 0.60 CYP2C9 (0.50) HSD11B1OPRM1CYP3A4CYP2C19
SCHEMBL8005872 0.60 MAOB (0.39) HSD11B1MAOBMAOA
SCHEMBL613615 0.60 OPRM1 (0.45) POLBOPRM1KCNH2TACR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414332-A1 ACRYLAMIDE COMPOUNDS AND THE USE THEREOF Shionogi & Co., Ltd. (JP) 2012-02-08 EP disclosed
WO-2010114181-A1 ACRYLAMIDE COMPOUNDS AND THE USE THEREOF SHIONOGI & CO., LTD. (JP) 2010-10-07 WO disclosed