SCHEMBL5397952

SCHEMBL5397952

Fc1cc2nc(SCCN3CCNCC3)[nH]c2cc1F

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.58
TSHR P16473 1/20 0.58
RAB9A P51151 2/20 0.55
NPC1 O15118 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
OPRL1 P41146 14/20 0.52
TNKS O95271 1/20 0.43
PARP1 P09874 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
GRIN2A Q12879 1/20 0.43
GRIN2B Q13224 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14502993 0.90 ALDH1A1 (0.67) ALDH1A1TSHRRAB9ANPC1SMN1; SMN2
Trifluoroacetic Acid SCHEMBL1704549 0.90 ALDH1A1 (0.49) ALDH1A1TSHRRAB9ANPC1SMN1; SMN2
SCHEMBL5381229 0.85 ALDH1A1 (0.53) ALDH1A1TSHRRAB9ANPC1SMN1; SMN2
SCHEMBL5381243 0.85 ALDH1A1 (0.53) ALDH1A1TSHRRAB9ANPC1SMN1; SMN2
SCHEMBL5387405 0.83 ALDH1A1 (0.57) ALDH1A1TSHRRAB9ANPC1SMN1; SMN2
SCHEMBL14502995 0.79 ALDH1A1 (0.80) ALDH1A1TSHRRAB9ANPC1SMN1; SMN2
SCHEMBL1704979 0.79 RAB9A (0.74) ALDH1A1TSHRRAB9ANPC1SMN1; SMN2
Hydrochloric Acid SCHEMBL1704951 0.78 RAB9A (0.73) TSHRRAB9ANPC1SMN1; SMN2TNKS
Trifluoroacetic Acid SCHEMBL5384259 0.77 ALDH1A1 (0.45) ALDH1A1TSHRRAB9ANPC1SMN1; SMN2
Trifluoroacetic Acid SCHEMBL5384262 0.77 ALDH1A1 (0.45) ALDH1A1TSHRRAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1642899-B1 2,4-BIS(TRIFLUOROETHOXY)PYRIDINE COMPOUND AND MEDICINE CONTAINING THE SAME KOWA CO (JP) 2012-08-15 EP disclosed
US-7223764-B2 2,4-bis (trifluoroethoxy)pyridine compound and drug containing the compound KOWA CO., LTD. (JP) 2007-05-29 US disclosed
EP-1642899-A1 2,4-BIS(TRIFLUOROETHOXY)PYRIDINE COMPOUND AND MEDICINE CONTAINING THE SAME Kowa Co., Ltd. (JP) 2006-04-05 EP disclosed
US-20050020606-A1 2,4-Bis (trifluoroethoxy)pyridine compound and drug containing the compound KOWA CO., LTD. (JP) 2005-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020606-A1 2,4-Bis (trifluoroethoxy)pyridine compound and drug containing the compound ACAT2, ACAT1, CYP7A1 ALDH1A1 586/4885TSHR 3355/4885RAB9A 855/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.