SCHEMBL5403418

SCHEMBL5403418

O=C(O)CCN(CCc1ccc(Cl)cc1Cl)C(=O)c1ccccc1-c1ccccc1C(=O)NCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.47
CHRNB4 P30926 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA4 P43681 1/20 0.47
HPGD P15428 3/20 0.47
LMNA P02545 2/20 0.47
ALDH1A1 P00352 1/20 0.47
PLAAT3 P53816 1/20 0.46
PLAAT5 Q96KN8 1/20 0.46
PLAAT2 Q9NWW9 1/20 0.46
PLAAT4 Q9UL19 1/20 0.46
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
CNR1 P21554 2/20 0.43
KCNA5 P22460 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HSP90AA1 P07900 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4930717 0.97 ALDH1A1 (0.48) CHRNB2CHRNB4CHRNA3CHRNA4HPGD
SCHEMBL5409628 0.95 HPGD (0.44) CHRNB2CHRNB4CHRNA3CHRNA4HPGD
SCHEMBL5399392 0.94 ALDH1A1 (0.45) CHRNB2CHRNB4CHRNA3CHRNA4HPGD
SCHEMBL5395356 0.94 KMT2A (0.44) CHRNB2CHRNB4CHRNA3CHRNA4HPGD
SCHEMBL5392441 0.92 HPGD (0.45) CHRNB2CHRNB4CHRNA3CHRNA4HPGD
SCHEMBL5408418 0.92 CNR1 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4HPGD
SCHEMBL5397846 0.92 MEN1 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4HPGD
SCHEMBL5409616 0.91 PLAAT3 (0.53) HPGDLMNAPLAAT3PLAAT5PLAAT2
SCHEMBL5404255 0.91 L3MBTL1 (0.47) HPGDALDH1A1PLAAT3PLAAT5PLAAT2
SCHEMBL5404133 0.91 HTT (0.54) HPGDLMNAALDH1A1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7285680-B2 β-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-10-23 US disclosed
US-20050256160-A1 Beta-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2005-11-17 US disclosed
EP-1533294-A1 BETA-ALANINE DERIVATIVE AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2005-05-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050256160-A1 Beta-alanine derivatives and the use thereof TGFB1, PML, APOB CHRNB2 857/4885CHRNB4 989/4885CHRNA3 1766/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.